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7084117 Pharmaceutical compositions which inhibit vascular proliferation and method of use thereof  
The present invention relates to a method of treating vascular proliferation in a patient in need thereof. The method includes the step of administering a therapeutically effective amount of a...
7067490 Hepta-, Octa-and nonapeptides having antiangiogenic activity  
Compounds of formula (SEQ ID NO:1), which are useful for treating conditions that arise from or are exacerbated by angiogenesis, are described. Also disclosed are pharmaceutical compositions...
7067489 Hematopoietic stimulation  
Methods and products for stimulating hematopoiesis, preventing low levels of hematopoietic cells and producing increased numbers of hematopoietic and mature blood cells are provided. The methods...
7063842 Compounds and methods for inhibiting the interaction between α-catenin and β-catenin  
Modulating agents for inhibiting an interaction between α-catenin and β-catenin are provided. The modulating agents comprise one or more of: (a) a β-catenin HAV motif; (b) a peptide analogue or...
7060670 Stereoselective antifibrillogenic peptides and peptidomimetics thereof  
The present invention relates to antifibrillogenic agents for inhibiting amyloidosis and/or for cytoprotection for the treatment amyloidosis disorders. These agents include peptides, isomers...
7053054 Purified LH  
A process for the purification of recombinant human Luteinizing Hormone (LH) from a sample of crude recombinant LH in the supernatant of CHO cells comprises the combined use of the ion-exchange...
7052703 T-cell receptorγ alternate reading frame protein, (TARP) and uses thereof  
This invention provides nucleic acids containing sequences from a TCRγ transcript from prostate epithelial cells and many breast cancer cells and a T-cell receptor gamma Alternate Reading frame...
7037897 TRI-, TETRA-, and penta-peptides having antiangiogenic activity  
Compounds of formula (SEQ ID NO:1), which are useful for treating conditions that arise from or are exacerbated by angiogenesis, are described. Also disclosed are pharmaceutical compositions...
7034002 Angiotensin converting enzyme inhibitor  
The present invention provides an angiotensin converting enzyme inhibitor having strong activity of inhibiting angiotensin converting enzyme, good hue and easily to take in which is a composition...
7034003 Somatostatin and somatostatin agonists for decreasing body weight  
The present invention relates to a method of decreasing body weight in a patient. The method includes the step of administering a therapeutically effective amount of a somatostatin or a...
7033794 Basolateral sorting signal and inhibitors thereof  
Mono-leucine dependent basolateral sorting signal consisting of the amino acid sequence X 1 h 2 X 3 h 4 L p 5 p 6 , wherein: X 1 represents a polar amino acid residue or alanine, h 2 represents...
7026289 Method and compositions for treating hyperlipidemia and other conditions  
The present invention relates to a method of treating hyperlipidemia and to reducing triacylglycerols, glycerol and cholesterol in a patient. The method includes the step of administering a...
7026296 Methods of treating dry eye disorders  
Inhibitors of cytokine synthesis in nonimmune, resident ocular surface cells are useful for treating dry eye disorders and other disorders requiring the wetting of the eye.
7022675 Wound healing compositions  
Methods and compositions based on chemical analogs of angiotensin II and analogs of angiotensin II fragments useful for accelerating wound healing in mammals.
7005418 Method for the therapeutic management of extrauterine proliferation of endometrial tissue, chronic pelvic pain and fallopian tube obstruction  
The present inventions provides a method for therapeutic management of extrauterine proliferation of endometrial tissue, chronic pelvic pain and fallopian tube obstruction by short term induction...
7005420 Ionic molecular conjugates of N-acylated derivatives of poly(2-amino-2-deoxy-D-glucose) and polypeptides  
A copolymer comprising an N-acylated derivative, and a composition comprising said copolymer and a polypeptide, said polypeptide comprising at least one effective ionogenic amine, wherein at least...
6992063 Compositions and method for regulating apoptosis  
Peptides and peptidomimetics capable of modulating apoptosis through their interaction with cellular IAPs (inhibitor of apoptosis proteins) are disclosed. The peptides and mimetics are based on the...
6989371 Bombesin analogs for treatment of cancer  
The present invention encompasses novel peptides that are antagonists to bombesin and bombesin like peptides and are useful in the treatment of cancer. The invention particularly relates to the...
6982249 Bradykinin analogs as selective inhibitors of cell activation  
The present invention provides bradykinin peptide analogs, compositions, and methods of inhibiting thrombin-induced platelet and other cell activation. The bradykinin analogs comprise single or...
6967192 Seventeen amino acid peptide (Peptide P) for treating ischemia and reperfusion injury  
Peptide P, having the amino acid sequence Tyr-D-Ala-Phe-Ala-Asp-Val-Ala-Ser-Thr-Ile-Gly-Asp-Phe-His-Se r-Ile-NH2-SEQ ID NO:1, is useful to treat ischemia.
6964948 Therapeutic peptide-based constructs derived from Domain II of bactericidal/permeability-increasing protein  
The present invention relates generally to small peptide-based constructs, including derivatized constructs, and their therapeutic uses. The constructs and derivatized constructs can have at least...
6962904 Elastin peptide analogs and uses thereof  
The present invention is directed to a composition which is used to enhance the elasticity and/or appearance of tissue. Specifically, the present invention is directed to a composition formulated...
6953779 Melanocortin receptor antagonists and modulations of melanocortin receptor activity  
The clinical outcome of disseminated melanoma is grim. Small molecular weight antagonists (preferably about seven amino acid residues) specific for MCR on melanoma cells are provided for the...
6951652 Vaccine for prevention of gram-negative bacterial infections and endotoxin related diseases  
A vaccine is disclosed which is useful for protecting a host from Gram negative infections and the effects of endotoxin, therefore preventing sepsis and septic shock. The vaccine is prepared by...
6951843 Peptide derivatives and their pharmaceutically acceptable salts, thereof, processes for preparation of both and use thereof  
The present invention provides a peptide derivative of formula (I) wherein X is —CHOH— or —CO—; R 1 and R 2 are hydrogen or substituted oxycarbonyl; R 3 is substituted oxycarbonyl;...
6949513 Polypeptides of covalently linked synthetic bioactive peptide analog(s) for treatment of cancer  
A polypeptide of the formula (I), P a -L-P b -L-P c -L-P d .
6939847 Use of colostrinin, constituent peptides thereof, and analogs thereof, as oxidative stress regulators  
The present invention provides methods that utilize compositions containing colostrinin, an constituent peptide thereof, an active analog thereof, and combinations thereof, as an oxidative stress...
6936587 Anti-invasive and anti-angiogenic compositions  
A peptide compound having the sequence Lys-Pro-Ser-Ser-Pro-Pro-Glu-Glu [SEQ ID NO:2] or a substitution variant, addition variant or other chemical derivative thereof inhibits cell invasion,...
6913761 Bioimplant formulation  
A pharmaceutical and/or veterinary formulation comprising about 2-30% (w/w) (on an active basis) of at least one active agent, about 0.5-20.0% (w/w) of a pore-foaming agent and the balance stearin....
6914048 Method for delivery of molecules to intracellular targets  
Disclosed are β-peptides and β-peptide conjugates that are capable of diffusing or otherwise being transported across the cell membranes of living cells. The β-peptides contain at least six...
6906037 Therapeutic peptide-based constructs  
The present invention relates generally to small peptide-based constructs and their therapeutic uses. The sequences of these peptide-based constructs are based on a reverse subsequence derived from...
6903074 Neuromedin b and somatostatin receptor agonists  
A novel class of analogs which exhibit both high affinity and selectivity for Neuromedin B and Somatostann receptors are claimed. One example is Nal-Tyr-cyclo(D-Cys-D-Trp-Lys-D-Cys)-Abu-Nal-NH 2 .
6900176 Pest control agents/depsipeptides  
The present invention relates to the use of 24-membered cyclodepsipeptides of the formula (1) in which R 1 and R 2 are as defined in the description, for controlling animal pests in...
6893645 Process to make a sustained release formulation  
This invention pertains to a process for making a sustained release complex. Compound (I), which comprises Compound (A), having formula (A), and a copolymer comprising poly...
6890902 Cytotoxic modified lactoferrin peptides  
The present invention provides a modified lactoferrin peptide which is cytotoxic, 7 to 25 amino acids in length, with three or more cationic residues and which has one or more extra bulky and...
6878689 Preventives or remedies for heart failure  
Preparations for preventing or treating acute heart failure, chronic heart failure at a phase of acute exacerbation or heart failure at a phase of transition to chronic heart failure, which contain...
6875743 Cell adhesion inhibitors  
The present invention relates to novel compounds that are useful for inhibition and prevention of cell adhesion and cell adhesion-mediated pathologies. This invention also relates to pharmaceutical...
6875744 Short bioactive peptides  
Short bioactive peptides containing phenylalanine, leucine, alanine, and lysine residues are disclosed. The peptides can be used in antibacterial, antifungal, anticancer, and other biological...
6866848 Antigenic polypetide sequence of factor VIII, fragments and/or epitopes there of  
An antigenic polypeptide of factor VIII comprises a polypeptide included between the Glutamic Acid 1649 and Asparagine 2019, preferably between Arginine 1652 and Arginine 1917 of the polypeptide of...
6864239 Methods and compounds for prevention and treatment of elevated intraocular pressure and related conditions  
A GPCR-like protein is described, as well as inhibitory/antagonistic compounds and compositions comprising such inhibitors/antagonists of the protein. Such compounds may be used for treating...
6858210 Therapeutic and diagnostic domain 1 β2GPI polypeptides and methods of using same  
The present invention provides domain 1 β 2 GPI polypeptides, polynucleotides encoding these polypeptides, mimetics of these polypeptides, and methods using domain 1 β 2 GPI polypeptides and...
6858396 Positively charged non-natural amino acids, methods of making and using thereof in peptides  
This invention relates to positively charged non-natural amino acids, methods of making thereof, and utilization thereof in peptides.
6855692 Histogranin peptides and their analgesic use  
The invention relates to linear and cyclic peptide and pseudopeptide compounds useful as analgesics, pharmaceutical compositions comprising such compounds, the use of the compounds and the...
6855695 Water-soluble SHPs as novel alkylating agents  
The present invention relates to compounds according to the structure (I): Where R is —CH 3 or —CH 2 CH 2 Cl; R′ is C 1 -C 7 alkyl or —CH 2 CH 2 Cl; R 2 or R 4 is OPO 3 H 2 , NO 2...
6852688 Compositions for treating diabetic retinopathy and methods of using same  
The subject invention provides novel methods and materials for treating diabetic retinopathy. One embodiment of the subject invention involves the co-administration of a somatostatin, or analogue...
6852695 Orally active fraction of momordica charantia, active peptides thereof, and their use in the treatment of diabetes  
A water soluble extract of M.charantia named MC6, methods for its preparation and methods for its use in the treatment of hyperglycemic disorders are provided. The active MC6 is characterized by...
6852321 Lectin-derived progenitor cell preservation factor and methods of use  
The invention relates to an isolated nucleic acid molecule that encodes a protein that is effective to preserve progenitor cells, such as hematopoietic progenitor cells. The nucleic acid comprises...
6852685 Use of colostrinin, constituent peptides thereof, and analogs thereof to promote neuronal cell differentiation  
The present invention discloses a use of colostrinin, a constituent peptide thereof, and/or an analog thereof as a neural cell regulator in animals including humans.
6852697 Peptides for treatment of inflammation and shock  
Submandibular peptides have been isolated and characterized and provide pharmaceutical compositions for the treatment or prevention of anaphylactic reactions, endotoxic reactions and SIRS-induced...
6844318 Peptidase-cleavable, targeted antineoplastic drugs and their therapeutic use  
This invention is directed to antineoplastic agents conjugated to enzyme-cleavable peptides comprising the amino acid recognition sequence of a membrane-bound and/or cell-secreted peptidase, and to...