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5425943 Modified tPA-containing injection composition having increased solubility  
An injection composition comprises a pharmacologically effective amount of a modified tPA, 47.5 mM or more of an amino acid or a salt thereof and is improved in view of stability and solubility.
5425942 Polyfunctinal protease  
The present invention provides a human polyfuctional protease chracterized in that the protease has unique enzymological and physicochemical properties:
5413786 Method of accelerating blood coagulation using a metal complex of oxidized ellagic acid  
Blood coagulation is accelerated by contacting blood with an accelerator of hydrolase activity. The activation of the precursors of serine protease including Factor XII and the enzyme activity of...
5411885 Methods for tissue embedding and tissue culturing  
Methods of embedding and culturing tissue employing a fibrin glue composition of 2 to 100 mg/ml fibrinogen, 1 to 200 U/ml fibrinogen-activating enzyme, and 1 to 30 mM Ca(II) compound, are disclosed.
5409700 Pharmaceutical compositions comprising modified and unmodified plasminogen activators  
The present invention relates to pharmaceutical compositions comprising a combination of two different plasminogen activators which are used for the prophylaxis and therapie of thrombosis.
5409699 Compositions containing glycosylated molecules having human tissue type plasminogen activator enzymatic activity  
The invention is a pharmaceutical composition containing a glycosylated protein having human tissue type plasminogen activator activity of at least 1.4 MU/ml, citrate, and at least one of a number...
5407673 Fibrinolysis and fibrinogenolysis treatment  
Disclosed is a fibrinolysis and fibrinogenolysis treatment which includes parenterally introducing into the body of a human patient human plasmin in fibrinolytically and fibrinogenolytically active...
5405607 Method for preparing fibrinogen adhesive from whole blood  
A process and apparatus for one-step preparation of the fibrinogen component of an adhesive is described. The fibrinogen is precipitated directly from plasma using polyethylene glycol. This permits...
5397704 Ultra-pure thrombin preparation  
An ultra-pure, clear thrombin solution having a high specific activity is described as well as a method of manufacture.
5393666 Method of activating prothrombin  
There is disclosed a method of activating prothrombin by means of trypsin, wherein the prothrombin is recovered from a blood or plasma fraction, treated with trypsin immobilized on a...
5391371 Use of an enzyme containing granulate in a method for production of a pelletized fodder  
An enzyme containing T-granulate, coated with a coating agent comprising a high melting fat or wax, is combined with a mixture containing fodder components, and the combination is steam treated and...
5389538 Mutant human prourokinase  
A mutant human prourokinase wherein a neutral amino acid in the epidermal growth factor (EGF) region of human prourokinase (human PUK) has been replaced with a basic amino acid, or an acidic amino...
5385732 Variants of tissue plasminogen activator, compositions and methods of use for same  
A fibrinolytically active amino acid sequence variant of a plasminogen activator is prepared that has one or more glycosylation sites in regions that are not glycosylated in the native molecule....
5376633 Method for deactivating viruses in blood component containers  
The present invention provides a method for inhibiting viral proliferation by preventing or inhibiting viral replication or killing the viruses on contact. Viral replication is prevented or...
5372812 Composition and method for acceleration of clot lysis  
The present invention relates to a novel treatment for blood clots within a patient or myocardial infarction which comprises administering a hapten-binding molecule capable of preventing inhibition...
5366869 Multiple coagulation test device and method  
A multiple coagulation test device has a plurality of tubes, each tube having associated coagulation detection means, and containing a treatment dosage of a coagulation enhancing agent. Whole blood...
5366730 Stabilized compositions having human tissue type plasminogen activator enzymatic activity  
Pharmaceutical preparation of a protein with t-PA activity with an enzymatic activity of at least 0.25 MU/ml. and a pH value of 4.5 to 9 which contains a substance of the group citric acid,...
5364622 Methods for preventing adhesions to organs and parts of organs by application of tissue plasminogen activator and hydroxyethylcellulose hydrogel  
A method for the prevention of adhesions to body organs and parts of organs caused by therapeutic intervention by applying a pharmaceutical composition of tissue plasminogen activator and an...
5352453 Compositions containing non-glycosylated human tissue type plasminogen activator  
Pharmaceutical compositions containing non-glycosylated human tissue type plasminogen activator (t-PA) having enzymatic activity of at least 0.1 MU/ml are disclosed. The compositions have a pH of...
5352452 Stabilized compositions containing non-glysylated human tissue type plasminogen activator derivative K2P pro  
Stabilized compositions containing a non-glycosylated human tissue type plasminogen activator derivative are disclosed. The derivative is referred to as K2P pro. The composition has enzymatic...
5350578 Inhibition of arterial thrombotic occlusion or thromboembolism  
The method of preventing arterial thrombotic occlusion or thromboembolism by administering plasma-derived or recombinant produced protein C alone or in combination with a thrombolytic agent or...
5342616 Method of administering tissue plasminogen activator  
The use of bolus injections of t-PA in the treatment of human beings with a thrombotic disorder.
5338546 Tissue plasminogen activator variants with decreased clearance  
Biologically active tissue plasminogen activator (t-PA) variants with decreased clearance as compared to wild-type t-PA are prepared, including variants that have one or more amino acid alterations...
5336495 Use of staphylokinase for the preparation of a pharmaceutical composition for treating arterial thromboisi  
The present invention relates to the use of staphylokinase for the preparation of a pharmaceutical composition for treating arterial thrombosis, such as e.g. myocardial infarction. It is...
5334384 Process for purification of streptakinase using a reducing agent  
A process for the separation of streptokinase from contaminating proteins in a streptokinase-containing mixture, which comprises treating the mixture with a reducing agent to reduce disulphide...
5326562 Pharmaceutical dosage unit for treating inflammation comprising protease nexin-I  
Methods and pharmaceutical compositions for treatment of inflammation and arthritis using protease nexin-I as an active ingredient are disclosed.
5324647 Fibrin coated polymer surfaces  
Surfaces of polymeric materials are coated with a layer of thermally denatured fibrinogen. The fibrinogen may be treated with thrombin to produce fibrin, and additional fibrinogen and factor XIII...
5324514 Compositions of digestive enzymes and salts of bile acids and process for preparation thereof  
Disclosed are gastric acid-resistant polymer-coated digestive enzymes/ursodeoxycholate compositions, process for their preparations and methods of treating digestive disorders, treating impaired...
5316766 Thrombosis treatment with fibrinolytics and prostacyclins  
The combination of a fibrinolytic and a prostacyclin analogue is very useful for thrombosis treatment, especially to avoid subsequent rethrombosis.
5315998 Booster for therapy of diseases with ultrasound and pharmaceutical liquid composition containing the same  
A booster comprising a plenty of microbubbles of a gas in a liquid, e.g. about 4×10 7 cells/ml of microbubbles of a gas having a diameter of 0.1 to 100 μm in a 3 to 5% human serum albumin...
5308617 Protein heparin conjugates  
A pharmaceutical composition is prepared wherein a biologically active conjugated protein is selectively conjugated to at least one heparin fragment having a terminal 2,5-anhydro-D-mannose residue...
5304383 Pharmaceutical preparation based on Lys-plasminogen  
There is disclosed a pharmaceutical preparation based on Lys-plasminogen and available in the lyophilized form. This preparation contains a serine-protease inhibitor and optionally an inhibitor...
5304372 Process for preparing a human thrombin concentrate intended for therapeutic use  
Process for preparing a human thrombin concentrate from the PPSB fraction of plasma that does not involve any addition of factors of animal origin to induce activation of the prothrombin to produce...
5302390 Hybrid proteins of human plasminogen and human t-PA, pharmaceutical compositions and methods of treatment  
A hybrid plasminogen activator which comprises the five kringle domains of plasminogen linked to the B-chain of t-PA or u-PA via an amino acid sequence comprising, respectively, the t-PA cleavage...
5298255 Antithrombic medical material, artificial internal organ, and method for production of antithrombic medical material  
An antithrombic medical material, having superposed on the surface of a substrate formed of a polymer material a polymerized protein substantially free at least from erythrocyte and leukocyte, a...
5296223 Subtilisin as an oral thrombolytic agent  
There are provided thrombolytic agents suited for oral administration. The agent comprises a proteolytic enzyme of subtilisin family, such as subtilisin BPN', subtilisin Carsberg, subtilisin...
5296357 Method for the detection of plasminogen activators, their inhibitors of stimulators  
The invention relates to a method for the detection of the functional activity of plasminogen activators and of their inhibitors and stimulators in biological samples, and to reagents for this method.
5290552 Surgical adhesive material  
The present invention provides a surgical adhesive comprising, in an aqueous composition, fibrinogen, FXIII, collagen, thrombin, Ca 2 + and optionally, an antifibrinolytic agent. The present...
5288490 Thrombus-targeted complexes of plasminogen activator and fibrin fragments  
Thrombolytic hybrids are formed as covalent or non-covalent complexes of fibrin fragments and plasminogen activator molecules. Native plasmin degradation fragments of fibrin or non-native fibrin...
5278144 Antithrombosis agents  
Analogs of Factor Xa (Factor Xai) which are inactive as proteases in the prothrombinase reaction are useful in treatment of diseases characterized by thrombosis. These antithrombotic agents can be...
5275946 Thrombolytic agents with modified kringle domains  
This invention relates to analogs of thrombolytic agents having a modified kringle domain. More specifically, this invention is directed to TPA type compounds wherein modifications occur in the...
5272076 Compounds and methods for treatment of thromboembolic disorders using an adduct of t-PA  
The present invention provides adducts of human t-PA derivatives, which comprise a t-PA derivative that lacks the Finger, Growth Factor and Kringle 1 domains, bound to an amphipathic molecule. The...
5270040 Vectors and compounds for expression of human protein C  
The present invention comprises novel DNA compounds which encode human protein C activity. A variety of eukaryotic and prokaryotic recombinant DNA expression vectors have been constructed that...
5258180 Tissue plasminogen activator having fibrin specific properties and deletion of amino acids 466-970, compositions and methods of treatment  
A tissue plasminogen activator (t-PA) variant is prepared that has an amino acid deletion at positions 466 to 470 of the corresponding wild-type t-PA. This alteration renders the variant fibrin...
5256642 Compositions of soluble complement receptor 1 (CR1) and a thrombolytic agent, and the methods of use thereof  
The present invention relates to compositions comprising soluble complement receptor 1 (CR1) and a thrombolytic agent. In a specific embodiment, the thrombolytic agent is anisoylated human...
5252463 Clipsin, a chymotrypsin-like protease and method of using same  
A novel M r 25,000 chymotrypsin-like protease, termed clipsin, which binds to a-1-AChy in a sodium dodecyl sulfate-resistant manner, preferentially degrades β-APP, and shows high activity for a...
5244676 Modified tissue plasminogen activator with modified glycosylation site  
A modified t-PA having improved in vivo half-life is disclosed comprising in sequence a fibronectin finger-like domain F, a growth factor domain GF, a sequence of two K2 kringle regions and a...
5244673 Medicamentous form for use as an ophthalmologic, otolaryngologic, or dermatologic drug  
A medicamentous form or composition with antiexudation, antiphlogistic, and antimicrobial effects in an aqueous or ointment base, suitable above all as an ophthalmologic, otolaryngologic, or...
5242688 Method of treating thromboembolic disorders by administration of diglycosylated t-PA variants  
The present invention provides a method of treating thromboembolic disorders with the diglycosylated form of a tissue plasminogen activator derivative that lacks the Finger, EGF and Kringle I...
5240845 Mutated streptokinase proteins  
This invention relates to a novel chemically synthesized gene including a base sequence coding for the primary amino acid sequence of natutal-type streptokinase, a corresponding plasmid...