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US20090264289 |
Use of Arylcarboxylic Acid Biphenylamides for Seed Treatment
The invention relates to the use of arylcarbonic acid biphenylamides of formula (I)
wherein
X is halogen or methyl; n is zero, 1 or 2; Y is cyano, nitro, halogen, C 1 -C 4 -alkyl, C 1 -C 4...
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US20090258912 |
N-(1-Alkyl-2-Phenylethyl)-Carboxamide Derivatives and Use Thereof as Fungicides
A compound of general formula (I):
A process for preparing this compound. A fungicidal composition comprising a compound of general formula (I). A method for treating plants by applying a...
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US20090258887 |
Novel Carboxylic Acid Derivatives
The present invention is concerned with novel arylalkyl carboxylic acid derivatives, more specifically, with acylates of arylalkyl carboxylic acids with naturally occurring, non-toxic hydroxy,...
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US20090227563 |
HERBICIDAL COMPOSITIONS HAVING IMPROVED EFFECT
The present invention concerns boosting the activity of crop protection materials comprising active ingredients from the class of the phenyl-substituted cyclic ketoenols through the addition of...
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US20090221651 |
CHEMICAL PRECONDITIONING AS A PREVENTATIVE OR TREATMENT FOR EXCITOTOXIC SYNAPTIC DAMAGE
A method of preventing HIV-1 associated dendritic pathology in a brain cell, comprising contacting the cell with a therapeutically effective dose of a mitochondrial ATP-sensitive potassium channel...
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US20090215838 |
ORGANIC NITRIC OXIDE ENHANCING SALTS OF ANGIOTENSIN II ANTAGONISTS, COMPOSITIONS AND METHODS OF USE
The invention describes compositions and kits comprising at least one organic nitric oxide enhancing salt of an angiotensin π antagonist, and, optionally, at least one nitric oxide enhancing...
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US20090197924 |
2-AMINO-2-PHENYL-ALKANOL DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
2-amino-2-phenyl-alkanol ester derivatives of general formula (I) in which: R 1 is H, straight or branched 1 to 4C alkyl, straight or branched 2 to 4C alkyl substituted by OH, alkoxy, alkylthio,...
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US20090196906 |
Kinase inhibitors
The present invention relates to drug delivery systems comprising ocular implant, which include organic molecules, capable of modulating tyrosine kinase signal transduction in order to regulate,...
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US20090192172 |
2-Alkyl-Cycloalk(en)yl-Carboxamides
Novel 2-alkylcycloalk(en)ylcarboxamides of the formula (I)
in which
X, s, R 1 , L, R 2 and A are as defined in the description,
a plurality of processes for preparing these compounds...
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US20090156616 |
THERAPEUTIC AGENTS
The present invention relates to compounds of formula (I) and processes for preparing such compounds, their use in the treatment of obesity, psychiatric and neurological disorders, to methods for...
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US20090143445 |
HDAC Inhibitors
This invention provides the compound having the structure
wherein n is 1-10; X is C—R 11 or N, wherein R 11 is H, OH, SH, F, Cl, SO 2 R 7 , NO 2 , trifluoromethyl, methoxy, or CO—R 7...
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US20090143409 |
3-PYRIDINECARBOXAMIDE DERIVATIVES AS HDL-CHOLESTEROL RAISING AGENTS
The present invention relates to a method of raising HDL cholesterol comprising administering to a patient in need thereof a compound of the formula
wherein A, G, R 1 to R 8 and R 17 are as...
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US20090136592 |
Vitamin preparation
Two-phase preparation for temporally gradual administration comprising
a) a phase (A) comprising water soluble vitamins and/or the corresponding provitamins, wherein phase (A) does not...
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US20090130163 |
Drugs With Improved Hydrophobicity For Incorporation in Medical Devices
The invention provides a medical device comprising a hydrophobic analog of a medicament known to inhibit cell proliferation and migration. The invention also provides a method of treating a...
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US20090118340 |
Method for inhibiting and/or preventing formation of cancer metastases and seconddary malignant cancers
The invention relates to a method for inhibiting and/or preventing formation of cancer metastases and secondary malignant cancers by administration to a subject of an effective amount of a...
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US20090118225 |
1-Methyl Nicotinamide and Derivatives for Treatment of Gastric Injury
The present invention is directed to nicotinamide derivatives, and their use in treating gastrointestinal disorders.
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US20090105188 |
Compositions and Methods for Treating Necrotizing Enterocolitis
The present invention relates to a method for treating or preventing necrotizing enterocolitis (NEC) in a human neonate in need thereof, comprising administering to the neonate a pharmaceutically...
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US20090093525 |
Cyclopropyl aryl amide derivatives and uses thereof
Compounds of the formula:
wherein Ar 1 , Ar 2 , R 1 and R 2 are as defined herein. Also provided are pharmaceutical compositions, methods of using, and methods of preparing the subject compounds.
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US20090076095 |
DEUTERIUM-ENRICHED NICORANDIL
The present application describes deuterium-enriched nicorandil, pharmaceutically acceptable salt forms thereof, and methods of treating using the same.
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US20090075819 |
Indanyl- and Tetrahydronaphtyl-amino-thiourea Compounds for Combating Animal Pests
The present invention relates to Indanyl- and Tetrahydronaphtyl-amino-thiourea compounds of formula I
wherein the variables R 1 to R 4 are as in the description. The invention relates also to...
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US20090074884 |
FAMILY OF PFKFB3 INHIBITORS WITH ANTI-NEOPLASTIC ACTIVITIES
A methods and compounds for inhibiting 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3 (PFKFB3) are described. Also described are methods of inhibiting cell proliferation, treating cancer,...
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US20090054497 |
METHODS FOR ATTAINING ENHANCED SEXUAL WELLNESS USING ANHYDROUS COMPOSITIONS
The invention relates to a method of attaining enhanced sexual wellness of an individual comprising administering to the genital areas of the individual, an anhydrous composition comprising a...
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US20090054496 |
MICROBIOCIDES
The invention relates to a fungicidally active compound of the general Formula (I): where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently...
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US20090054372 |
Combination therapy for weight loss
The present invention is directed to methods and kits for achieving or maintaining weight loss. These kits and methods can include administering a pharmaceutical composition comprising phentermine,...
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US20090036495 |
Combinations Comprising Alpha-2-Delta Ligands and Ep4 Receptor Antagonists
The instant invention relates to a combination of an EP4-receptor antagonist and an alpha-2-delta ligand, and pharmaceutically acceptable salts thereof, pharmaceutical compositions thereof and...
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US20090036420 |
BENZAMIDE DERIVATIVES AND THEIR USE FOR TREATING CNS DISORDERS
The present invention relates to methods of treating CNS disorders with a compound of formula I
wherein
X, R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 , and R 8 are as defined in the...
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US20090028934 |
GRANULAR, GASTRO-RESISTANT PRODUCT BASED ON NIACIN OR DERIVATES THEREOF AND PROCESS FOR THE PRODUCTION OF SUCH A PRODUCT
A granular, gastro-resistant product based on niacin or derivatives thereof comprises an internal part in which the niacin is substantially concentrated and an external coating, provided to cover...
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US20090012130 |
Strategies for Designing Drugs that Target the Sir2 Family of Enzymes
The instant invention describes methods of identifying compounds that modulate the activity of Sir2 enzymes. Sir2 enzymes form a unique class Of NAD + dependent deacetylases required for diverse...
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US20090012126 |
Certain chemical entities, compositions, and methods
Chemical entities that modulate smooth muscle myosin and/or non-muscle myosin, and chemical entities, pharmaceutical compositions and methods of treatment of diseases and conditions associated with...
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US20080312295 |
Pesticidal Mixtures
Pesticidal mixtures comprising, as active components,
A) a phenylsemicarbazone compound of the formula (I),
where R 1 and R 2 are, independently of one another, hydrogen, cyano,...
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US20080311221 |
LEWIS ACID AND OIL-SOLUBLE HYBRID PESTICIDE CONCENTRATE THAT SPONTANEOUSLY FORMS A WATER-BASED MICROEMULSION
A chemically and physically stable, transparent, hybrid pesticide concentrate is provided for preparation of a water-based microemulsion formulation. The pesticides preferably comprise an...
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US20080311099 |
Pyridoxal-5-Phosphate and Related Compounds in Combination With Therapeutic Cardiovascular Compounds for Treating Angina
Methods for treating angina are described. A method for treating angina includes concurrently administering a compound with a therapeutic cardiovascular compound. A combination therapy employs...
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US20080293567 |
Fungicidal Mixtures Comprising Boscalid and Pyrimethanil
Fungicidal mixtures comprising
(1) boscalid of the formula (I)
and (2) pyrimethanil of the formula (II)
in a synergistically effective amount, methods for controlling harmful fungi using...
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US20080287499 |
N-DEACETYLTHIOCOLCHICINE DERIATIVES, THEIR USE AND PHARMACEUTICAL FORMULATIONS CONTAINING THEM
Disclosed is a series of N-deacetylthiocolchicine derivatives of formula I
in which:
the linker is a bivalent straight or branched C 1 -C 8 alkyl residue, C 3 -C 8 cycloalkyl, a...
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US20080287293 |
Pesticidal Mixtures
Pesticidal mixtures comprising, as active components,
1) an 1-arylpyrazole of the formula I
wherein R 1 is CN, C(═O)C 1 -C 4 -alkyl, or C(═S)NH 2 ; R 2 is S(O) n R 3 ; R 3 is C 1 -C 6...
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US20080279942 |
Pharmaceutical Preparation Containing an Angiotensin II Receptor Antagonist and a Calcium Channel Blocker
A pharmaceutical preparation comprising an angiotensin II receptor antagonist, a calcium channel blocker and at least one substance selected from the group consisting of a hydrophilic polymer, an...
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US20080269215 |
Bisamide Inhibitors of Hedgehog Signaling
The invention provides inhibitors of hedgehog signaling that are useful as a therapeutic agents for treating malignancies where the compounds have the general formula I:
wherein ring A, ring B,...
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US20080249140 |
Quaternary 3 -Amido, N-Methylpyridinium Salts as Anti-Inflammatory Agents
A novel group of anti-inflammatory compounds are salts composed of the anion of a nonsteroidal anti-inflammatory acid drug (NSAID) and the cation N(1)-methylnicotinamide, which both anion and...
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US20080234336 |
Synergistic Imazalil Combinations
The present invention relates to synergistic combinations of the antifungal agent imazalil and another antifungal agent selected from the group consisting of boscalid, cyproconazole,...
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US20080227831 |
FOOD EXTRACTS FOR TREATMENT OF LIPOPROTEIN ABNORMALITIES AND SKIN DISEASES AND SKIN DISORDERS
The present invention is directed to N-methylnicotinamide containing food extracts, and their use in treating lipoprotein abnormalities and skin diseases and disorders.
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US20080221172 |
Use of Quaternary Pyridinium Compounds for Vasoprotection and/or Hepatoprotection
The invention relates to a method for the treatment or prevention of diseases or conditions associated with vascular endothelium dysfunction or liver injury comprising the administration to a...
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US20080220104 |
Compositions for producing satiety
Long term weight loss can be achieved and maintained with a formulation of over-the-counter life-enhancing dietary supplements. One or more supplements stimulate the release of serotonin within the...
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US20080214616 |
Pyridine Derivatives as Dipeptedyl Peptidase Inhibitors
The present invention is directed to compounds of formula (I) or a pharmaceutically acceptable salt thereof; wherein A is (1); X is selected from CH, CF and N; R5 is selected from H, C 1 -C 6 ...
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US20080214532 |
Carboxanilides as Microbiocides
Compounds of the formula (I) in which the substituents are as defined in claim 1 are suitable for use as microbiocides.
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US20080207702 |
Use of Quaternary Pyridinium Salts as Vasoprotective Agents
The invention relates to the use of quaternary pyridium salts of formula (1) wherein R is NH 2 , CH 3 , or N(H)CH 2 OH group, and X is pharmaceutically acceptable counterion, for the preparation of...
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US20080199538 |
Compound to enhance lucid erotic dreams
A compound that contains herbal supplements to increase the frequency and lucidity of a person's erotic or sexual dreams. The compound can be used by anyone wishing to enhance their lucid erotic...
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US20080194627 |
Aryl substituted pyridines and the use thereof
This invention relates aryl substituted pyridines of Formula I:
or a pharmaceutically acceptable salt, prodrug or solvate thereof, wherein Ar and R 1 —R 4 are set in the specification. The...
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US20080171774 |
Nicotinanilides, Method for Production Thereof and Agents Comprising the Same for Prevention of Fungal Pests
The present invention relates to nicotinanilides of the formula I
in which:
n=0, 1, 2; m=2, 3; X 1 =F, chlorine; X 2 =halogen; Y=CN, NO 2 , C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl, methoxy or...
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US20080153824 |
Method for Controlling Fungal Diseases in Leguminous Plants
Method for controlling rust infections in leguminous plants by using orysastrobin, mixtures of orysastrobin and a fungicidally active compound II from the group of the azoles, acylalanines, amine...
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US20080153701 |
Fungicidal Mixtures
Fungicidal mixtures, comprising as active components
1) carbamate oxime ethers of the formula I,
in which X is N or CH,
and
2) at least one active compound II selected...
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